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Pelabresib Constellation Pharmaceuticals Inhibitor 0610 (CPI-0610) is an investigational oral BET inhibitor that targets transcriptional regulators involved in myelofibrosis (1). It modulates megakaryocyte differentiation, proliferation, and reduces proinflammatory cytokine expression via the Nuclear Factor kappa-light-chain (NF-κB) pathway (1). BE
Pelabresib as a Disease-Modifying Myelofibrosis Option

Pelabresib as a Disease-Modifying Myelofibrosis Option

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