
1w2 min read
Medical Article
Pelabresib Constellation Pharmaceuticals Inhibitor 0610 (CPI-0610) is an investigational oral BET inhibitor that targets transcriptional regulators involved in myelofibrosis (1). It modulates megakaryocyte differentiation, proliferation, and reduces proinflammatory cytokine expression via the Nuclear Factor kappa-light-chain (NF-κB) pathway (1). BE

Pelabresib as a Disease-Modifying Myelofibrosis Option
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